Possible Antifertility Agents Belonging to Substituted Indoles.
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چکیده
منابع مشابه
Synthesis of 2-phenyl-5-sulpha/substituted-3- substituted phenyl azo indoles used as antifertility agent
–A novel series of 2-phenyl-5-sulpha/substituted-3-phenyl substituted azo indoles have been synthesized and tested as an antifertility activity in mature albino mice. The tested compounds showed significant antifertility activity. Keywords––Synthesis, Antifertility activity, Indore, Azo indoles, chemical analysis.
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Intramolecular tin and sulfur mediated free-radical cyclizations between an aryl isonitfile and a pendant TMSsubstituted alkyne give 2,3-disubstituted indoles from 5-exo-dig cyclization and nucleophilic trapping of the resulting indolenine intermediate. © 1999 Elsevier Science Ltd. All fights reserved. In spite of the fact that Fischer first described their synthesis some 115 years ago, 1 the g...
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ژورنال
عنوان ژورنال: Biological and Pharmaceutical Bulletin
سال: 1993
ISSN: 0918-6158,1347-5215
DOI: 10.1248/bpb.16.36